Compile Data Set for Download or QSAR
maximum 50k data
Found 39 of affinity data for UniProtKB/TrEMBL: P48163
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405808(CHEMBL5279096)
Affinity DataIC50:  150nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177180(3-(4-(4-hydroxyphenyl)piperazin-1-yl)-1-phenylpyrr...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405811(CHEMBL5277536)
Affinity DataIC50:  150nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405806(CHEMBL5275653)
Affinity DataIC50:  170nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405803(CHEMBL5284469)
Affinity DataIC50:  180nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405807(CHEMBL5287773)
Affinity DataIC50:  180nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405802(CHEMBL5278951)
Affinity DataIC50:  200nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405809(CHEMBL5283020)
Affinity DataIC50:  210nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405800(CHEMBL5267207)
Affinity DataIC50:  220nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177180(3-(4-(4-hydroxyphenyl)piperazin-1-yl)-1-phenylpyrr...)
Affinity DataIC50:  220nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405805(CHEMBL5289840)
Affinity DataIC50:  270nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405801(CHEMBL5289950)
Affinity DataIC50:  340nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405810(CHEMBL5284610)
Affinity DataIC50:  420nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177175(1-benzyl-3-(4-(4-hydroxyphenyl)piperazin-1-yl)-1-p...)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177184(1-(3-chloro-4-methylphenyl)3-(4-(4-hydroxyphenyl)p...)
Affinity DataIC50:  560nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405804(CHEMBL5279230)
Affinity DataIC50:  630nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405798(CHEMBL5218866)
Affinity DataIC50:  940nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405818(CHEMBL5273550)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of spermidine synthase activity was evaluatedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405825(CHEMBL5286488)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against Dihydrofolate reductase in rat liverMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405822(CHEMBL5274945)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of spermidine synthase activity was evaluatedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405816(CHEMBL5291081)
Affinity DataIC50:  1.31E+3nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405824(CHEMBL5279589)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of spermine synthase activity in rat ventral prostrate was evaluatedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405823(CHEMBL5286064)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of spermine synthase activity in rat ventral prostrate was evaluatedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405812(CHEMBL5281297)
Affinity DataIC50:  1.50E+3nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405815(CHEMBL5278596)
Affinity DataIC50:  1.60E+3nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405819(CHEMBL5282439)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of spermine synthase activity in rat ventral prostrate was evaluated at 100 uMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405826(CHEMBL5290463)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity against Dihydrofolate reductase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405820(CHEMBL5270965)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of spermidine synthase activity was evaluatedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405817(CHEMBL5267542)
Affinity DataIC50:  2.37E+3nMAssay Description:Inhibition of spermidine synthase activity was evaluatedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177177(1-phenyl-3-(4-(3-(trifluoromethyl)phenyl)piperazin...)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405821(CHEMBL5281258)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of spermine synthase activity in rat ventral prostrate was evaluatedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177179(3-(4-(4-fluorophenyl)piperazin-1-yl)-1-phenylpyrro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177178(1-benzyl-3-(4-(3-hydroxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405797(CHEMBL5277143)
Affinity DataIC50:  1.03E+4nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50405799(CHEMBL5283717)
Affinity DataIC50:  1.38E+4nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177181(3-(4-(4-methoxyphenyl)piperazin-1-yl)-1-phenylpyrr...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177182(1-benzyl-3-(4-(4-methoxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177183(1-(2,3-dichlorophenyl)-3-(4-(4-methoxyphenyl)piper...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50177176(1-benzyl-3-(4-(2-hydroxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed